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1

Bis(guanidinium) Receptors as Ribonuclease Active-Site Model Systems: Structural Changes and Solvent Effects

Thorsten Oost, Anna Filippazzi, Markus Kalesse

Journal:

European Journal of Organic Chemistry

Year:

1997

Language:

english

File:

PDF, 819 KB

english, 1997

2

Regio- and diastereo-selectivity of the insertion of aldehydes into alkyne zirconocene complexes

Martin E. Maier, Thorsten Oost

Journal:

Journal of Organometallic Chemistry

Year:

1995

Language:

english

File:

PDF, 1.10 MB

english, 1995

3

Discovery of a potent and selective Bcl-2 inhibitor using SAR by NMR

Andrew M. Petros, Jeffrey R. Huth, Thorsten Oost, Cheol-Min Park, Hong Ding, Xilu Wang, Haichao Zhang, Paul Nimmer, Renaldo Mendoza, Chaohong Sun, Jamey Mack, Karl Walter, Sarah Dorwin, Emily Gramling

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.84 MB

english, 2010

4

Potent and selective oxindole-based vasopressin 1b receptor antagonists with improved pharmacokinetic properties

Thorsten Oost, Gisela Backfisch, Swati Bhowmik, Marcel M. van Gaalen, Hervé Geneste, Wilfried Hornberger, Wilfried Lubisch, Astrid Netz, Liliane Unger, Wolfgang Wernet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 473 KB

english, 2011

5

Potent, selective inhibitors of protein tyrosine phosphatase 1B

Zhili Xin, Thorsten K Oost, Cele Abad-Zapatero, Philip J Hajduk, Zhonghua Pei, Bruce G Szczepankiewicz, Charles W Hutchins, Steve J Ballaron, Mike A Stashko, Tom Lubben, James M Trevillyan, Mike R Jir

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 214 KB

english, 2003

6

Synthesis of RNAse active site model systems using a steroid template

Thorsten Oost, Markus Kalesse

Journal:

Year:

1997

Language:

english

File:

PDF, 951 KB

english, 1997

7

10.1038/35050006

Fesik, Stephen W., Liu, Zhihong, Sun, Chaohong, Olejniczak, Edward T., Meadows, Robert P., Betz, Stephen F., Oost, Thorsten, Herrmann, Julia, Wu, Joe C.

Journal:

Year:

2000

Language:

english

File:

PDF, 375 KB

english, 2000

8

Studies Leading to Potent, Dual Inhibitors of Bcl-2 and Bcl-xL

Oost, Thorsten K., Belli, Barbara A., Ding, Hong, Bruncko, Milan, Joseph, Mary K., Kunzer, Aaron, Martineau, Darlene, McClellan, William J., Mitten, Michael, Ng, Shi-Chung

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 755 KB

english, 2007

9

Design and synthesis of substrate-based inhibitors of botulinum neurotoxin type B metalloprotease

Thorsten Oost, Chanokporn Sukonpan, Matthias Brewer, Michael Goodnough, William Tepp, Eric A. Johnson, Daniel H. Rich

Journal:

Year:

2003

Language:

english

File:

PDF, 363 KB

english, 2003

10

Discovery of Potent Antagonists of the Antiapoptotic Protein XIAP for the Treatment of Cancer

Oost, Thorsten K., Sun, Chaohong, Armstrong, Robert C., Al-Assaad, Ali-Samer, Betz, Stephen F., Deckwerth, Thomas L., Ding, Hong, Elmore, Steven W., Meadows, Robert P., Olejniczak, Edward T., Oleksije

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 269 KB

english, 2004

11

Discovery and Structure−Activity Relationship of Antagonists of B-Cell Lymphoma 2 Family Proteins with Chemopotentiation Activity in Vitro and in Vivo

Wendt, Michael D., Shen, Wang, Kunzer, Aaron, McClellan, William J., Bruncko, Milan, Oost, Thorsten K., Ding, Hong, Joseph, Mary K., Zhang, Haichao, Nimmer, Paul M., Ng, Shi-Chung, Shoemaker, Alexande

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 343 KB

english, 2006

12

Discovery of Aminoglycoside Mimetics by NMR-Based Screening of Escherichia c oli A-site RNA

Yu, Liping, Oost, Thorsten K., Schkeryantz, Jeffrey M., Yang, Jianguo, Janowick, Dave, Fesik, Stephen W.

Journal:

Journal of the American Chemical Society

Year:

2003

Language:

english

File:

PDF, 256 KB

english, 2003

13

Structural Basis for BABIM Inhibition of Botulinum Neurotoxin Type B Protease

Hanson, Michael A., Oost, Thorsten K., Sukonpan, Chanokporn, Rich, Daniel H., Stevens, Raymond C.

Journal:

Journal of the American Chemical Society

Year:

2000

Language:

english

File:

PDF, 107 KB

english, 2000

14

Sequencing Hydroxyethylamine-Containing Peptides via Edman Degradation

Brewer, Matthias, Oost, Thorsten, Sukonpan, Chanokporn, Pereckas, Michael, Rich, Daniel H

Journal:

Organic Letters

Year:

2002

Language:

english

File:

PDF, 77 KB

english, 2002

15

Structural Basis for BABIM Inhibition of Botulinum Neurotoxin Type B Protease [ J. Am. Chem. Soc. 2000 , 122 , 11268−11269].

Oost, Thorsten K., Sukonpan, Chanokporn, Rich, Daniel H., Stevens, Raymond C.

Journal:

Journal of the American Chemical Society

Year:

2002

File:

PDF, 8 KB

2002

16

Design, synthesis and evaluation of MCH receptor 1 antagonists—Part II: Optimization of pyridazines toward reduced phospholipidosis and hERG inhibition

Roth, Gerald J., Heckel, Armin, Kley, Jörg T., Lehmann, Thorsten, Müller, Stephan G., Oost, Thorsten, Rudolf, Klaus, Arndt, Kirsten, Budzinski, Ralph, Lenter, Martin, Lotz, Ralf R.H., Schindler, Marcu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 277 KB

english, 2015

17

Design, synthesis and evaluation of MCH receptor 1 antagonists—Part III: Discovery of pre-clinical development candidate BI 186908

Oost, Thorsten, Heckel, Armin, Kley, Jörg T., Lehmann, Thorsten, Müller, Stephan, Roth, Gerald J., Rudolf, Klaus, Arndt, Kirsten, Budzinski, Ralph, Lenter, Martin, Lotz, Ralf R.H., Maier, Gerd-Michael

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 608 KB

english, 2015

18

Design, synthesis and evaluation of MCH receptor 1 antagonists—Part I: Optimization of HTS hits towards an in vivo efficacious tool compound BI 414

Müller, Stephan G., Heckel, Armin, Kley, Jörg T., Lehmann, Thorsten, Lustenberger, Philipp, Oost, Thorsten, Roth, Gerald J., Rudolf, Klaus, Arndt, Kirsten, Lenter, Martin, Lotz, Ralf R.H., Maier, Gerd

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.34 MB

english, 2015

19

Novel, potent, selective and brain penetrant vasopressin 1b receptor antagonists

Geneste, Hervé, Bhowmik, Swati, van Gaalen, Marcel M., Hornberger, Wilfried, Hutchins, Charles W., Netz, Astrid, Oost, Thorsten, Unger, Liliane

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2018

Language:

english

File:

PDF, 763 KB

english, 2018

20

Managing erosion of mangrove-mud coasts with permeable dams â lessons learned

Winterwerp, Johan C., Albers, Thorsten, Anthony, Edward J., Friess, Daniel A., MancheÃ±o, Alejandra GijÃ³n, Moseley, Kene, Muhari, Abdul, Naipal, Sieuwnath, Noordermeer, Joost, Oost, Albert, Saengsupa

Journal:

Ecological Engineering

Year:

2020

File:

PDF, 9.93 MB

2020